PDB Information

PDB3TJC
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of potent and highly selective thienopyridine janus kinase 2 inhibitors.
Schenkel, L.B., Huang, X., Cheng, A., Deak, H.L., Doherty, E., Emkey, R., Gu, Y., Gunaydin, H., Kim, J.L., Lee, J., Loberg, R., Olivieri, P., Pistillo, J., Tang, J., Wan, Q., Wang, H.L., Wang, S.W., Wells, M.C., Wu, B., Yu, V., Liu, L., Geuns-Meyer, S.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2011-08-24
Resolution2.400
CATH Insert Date04 Dec, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Dec, 2011 Chopped
B 05 Dec, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3tjcA01 07 Dec, 2011 3.30.200.20 Assigned
3tjcA02 07 Dec, 2011 1.10.510.10 Assigned
3tjcB01 07 Dec, 2011 3.30.200.20 Assigned
3tjcB02 07 Dec, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60674 JAK2_HUMAN Homo sapiens Tyrosine-protein kinase JAK2
O60674 JAK2_HUMAN Homo sapiens Tyrosine-protein kinase JAK2