PDB Information

PDB3SX0
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Bromo-deaza-SAH: a potent and selective DOT1L inhibitor.
Yu, W., Smil, D., Li, F., Tempel, W., Fedorov, O., Nguyen, K.T., Bolshan, Y., Al-Awar, R., Knapp, S., Arrowsmith, C.H., Vedadi, M., Brown, P.J., Schapira, M.
Bioorg. Med. Chem.
HeaderTransferase
Released2011-07-14
Resolution2.280
CATH Insert Date07 Aug, 2011

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Aug, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3sx0A01 12 Aug, 2011 1.10.260.60 Assigned
3sx0A02 12 Aug, 2011 3.40.50.150 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q8TEK3 DOT1L_HUMAN Homo sapiens Histone-lysine N-methyltransferase, H3 lysine-79 specific