PDB Information

PDB3SKC
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Pyrazolopyridine inhibitors of B-RafV600E. Part 2: structure-activity relationships.
Wenglowsky, S., Ahrendt, K.A., Buckmelter, A.J., Feng, B., Gloor, S.L., Gradl, S., Grina, J., Hansen, J.D., Laird, E.R., Lunghofer, P., Mathieu, S., Moreno, D., Newhouse, B., Ren, L., Risom, T., Rudolph, J., Seo, J., Sturgis, H.L., Voegtli, W.C., Wen, Z.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2011-06-22
Resolution3.200
CATH Insert Date21 Aug, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 22 Aug, 2011 Chopped
B 22 Aug, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3skcA01 26 Aug, 2011 3.30.200.20 Assigned
3skcA02 26 Aug, 2011 1.10.510.10 Assigned
3skcB01 25 Aug, 2011 3.30.200.20 Assigned
3skcB02 25 Aug, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf