PDB Information

PDB3QGY
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and structure-activity relationship of 3-aminopyrid-2-ones as potent and selective interleukin-2 inducible T-cell kinase (Itk) inhibitors
Charrier, J.D., Miller, A., Kay, D.P., Brenchley, G., Twin, H.C., Collier, P.N., Ramaya, S., Keily, S.B., Durrant, S.J., Knegtel, R.M., Tanner, A.J., Brown, K., Curnock, A.P., Jimenez, J.M.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2011-01-25
Resolution2.100
CATH Insert Date26 Jun, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 27 Jun, 2011 Chopped
B 27 Jun, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3qgyA01 29 Jun, 2011 3.30.200.20 Assigned
3qgyA02 29 Jun, 2011 1.10.510.10 Assigned
3qgyB01 28 Jun, 2011 3.30.200.20 Assigned
3qgyB02 28 Jun, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q08881 ITK_HUMAN Homo sapiens Tyrosine-protein kinase ITK/TSK
Q08881 ITK_HUMAN Homo sapiens Tyrosine-protein kinase ITK/TSK