PDB 3qgy
PDB Information
PDB | 3QGY |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Discovery and structure-activity relationship of 3-aminopyrid-2-ones as potent and selective interleukin-2 inducible T-cell kinase (Itk) inhibitors
J.Med.Chem.
|
Header | Transferase/Transferase Inhibitor |
Released | 2011-01-25 |
Resolution | 2.100 |
CATH Insert Date | 26 Jun, 2011 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 27 Jun, 2011 | Chopped |
B | 27 Jun, 2011 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
3qgyA01 | 29 Jun, 2011 | 3.30.200.20 | Assigned |
3qgyA02 | 29 Jun, 2011 | 1.10.510.10 | Assigned |
3qgyB01 | 28 Jun, 2011 | 3.30.200.20 | Assigned |
3qgyB02 | 28 Jun, 2011 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q08881 | ITK_HUMAN | Homo sapiens | Tyrosine-protein kinase ITK/TSK |
Q08881 | ITK_HUMAN | Homo sapiens | Tyrosine-protein kinase ITK/TSK |