PDB Information

PDB3O2M
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and characterization of non-ATP site inhibitors of the mitogen activated protein (MAP) kinases.
Comess, K.M., Sun, C., Abad-Zapatero, C., Goedken, E.R., Gum, R.J., Borhani, D.W., Argiriadi, M., Groebe, D.R., Jia, Y., Clampit, J.E., Haasch, D.L., Smith, H.T., Wang, S., Song, D., Coen, M.L., Cloutier, T.E., Tang, H., Cheng, X., Quinn, C., Liu, B., Xin, Z., Liu, G., Fry, E.H., Stoll, V., Ng, T.I., Banach, D., Marcotte, D., Burns, D.J., Calderwood, D.J., Hajduk, P.J.
Acs Chem.Biol.
HeaderTransferase/Inhibitor
Released2010-07-22
Resolution2.700
CATH Insert Date23 Jan, 2011

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 24 Jan, 2011 Chopped
B 24 Jan, 2011 Chopped
F 24 Jan, 2011 Rejected
G 24 Jan, 2011 Rejected

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3o2mA01 17 Feb, 2011 3.30.200.20 Assigned
3o2mA02 17 Feb, 2011 1.10.510.10 Assigned
3o2mB01 17 Feb, 2011 3.30.200.20 Assigned
3o2mB02 17 Feb, 2011 1.10.510.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P45983 MK08_HUMAN Homo sapiens Mitogen-activated protein kinase 8
Q9WVI9 JIP1_MOUSE Mus musculus C-Jun-amino-terminal kinase-interacting protein 1
Q9WVI9 JIP1_MOUSE Mus musculus C-Jun-amino-terminal kinase-interacting protein 1
P45983 MK08_HUMAN Homo sapiens Mitogen-activated protein kinase 8