PDB Information

PDB3MYG
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine Core.
Yu, T., Tagat, J.R., Kerekes, A.D., Doll, R.J., Zhang, Y., Xiao, Y., Esposite, S., Belanger, D.B., Curran, P.J., Mandal, A.K., Siddiqui, M.A., Shih, N.Y., Basso, A.D., Liu, M., Gray, K., Tevar, S., Jones, J., Lee, S., Liang, L., Ponery, S., Smith, E.B., Hruza, A., Voigt, J., Ramanathan, L., Prosise, W., Hu, M.
ACS Med Chem Lett
HeaderTransferase
Released2010-05-10
Resolution2.400
CATH Insert Date15 Aug, 2010

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3mygA01 15 Oct, 2010 3.30.200.20 Assigned
3mygA02 15 Oct, 2010 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14965 AURKA_HUMAN Homo sapiens Aurora kinase A