PDB 3lpb
PDB Information
PDB | 3LPB |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | Discovery and SAR of potent, orally available 2,8-diaryl-quinoxalines as a new class of JAK2 inhibitors
Bioorg.Med.Chem.Lett.
|
Header | Transferase |
Released | 2010-02-05 |
Resolution | 2.000 |
CATH Insert Date | 02 May, 2010 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 03 May, 2010 | Chopped |
B | 03 May, 2010 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
3lpbA01 | 21 Jul, 2010 | 3.30.200.20 | Assigned |
3lpbA02 | 21 Jul, 2010 | 1.10.510.10 | Assigned |
3lpbB01 | 21 Jul, 2010 | 3.30.200.20 | Assigned |
3lpbB02 | 21 Jul, 2010 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
O60674 | JAK2_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK2 |
O60674 | JAK2_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK2 |