PDB Information

PDB3KYR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Investigation of a-phenylnorstatine and a-benzylnorstatine as transition state isostere motifs in the search for new BACE-1 inhibiotrs
Wangsell, F., Nordeman, P., Savmarker, J., Emanuelsson, R., Jansson, K., Lindberg, J., Rosenqvist, A., Samuelsson, B., Larhed, M.
To be Published
HeaderHydrolase/Hydrolase Inhibitor
Released2009-12-07
Resolution2.600
CATH Insert Date23 Jan, 2011

PDB Images (10)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 24 Jan, 2011 Chopped
B 24 Jan, 2011 Chopped
C 24 Jan, 2011 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
3kyrA01 17 Feb, 2011 2.40.70.10 Assigned
3kyrA02 17 Feb, 2011 2.40.70.10 Assigned
3kyrB01 16 Feb, 2011 2.40.70.10 Assigned
3kyrB02 16 Feb, 2011 2.40.70.10 Assigned
3kyrC01 17 Feb, 2011 2.40.70.10 Assigned
3kyrC02 17 Feb, 2011 2.40.70.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P56817 BACE1_HUMAN Homo sapiens Beta-secretase 1
P56817 BACE1_HUMAN Homo sapiens Beta-secretase 1
P56817 BACE1_HUMAN Homo sapiens Beta-secretase 1
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