PDB 3k5k

PDB Information

PDB3K5K
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a 2,4-diamino-7-aminoalkoxyquinazoline as a potent and selective inhibitor of histone lysine methyltransferase G9a.
Liu, F., Chen, X., Allali-Hassani, A., Quinn, A.M., Wasney, G.A., Dong, A., Barsyte, D., Kozieradzki, I., Senisterra, G., Chau, I., Siarheyeva, A., Kireev, D.B., Jadhav, A., Herold, J.M., Frye, S.V., Arrowsmith, C.H., Brown, P.J., Simeonov, A., Vedadi, M., Jin, J.
J.Med.Chem.
HeaderTransferase
Released2009-10-07
Resolution1.700
CATH Insert Date15 Nov, 2009

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 15 Nov, 2009 Chopped
B 15 Nov, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3k5kA00 19 Aug, 2010 2.170.270.10 Assigned
3k5kB00 19 Aug, 2010 2.170.270.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q96KQ7 EHMT2_HUMAN Homo sapiens Histone-lysine N-methyltransferase EHMT2
Q96KQ7 EHMT2_HUMAN Homo sapiens Histone-lysine N-methyltransferase EHMT2