PDB Information

PDB3JYA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of 3H-benzo[4,5]thieno[3,2-d]pyrimidin-4-ones as Potent, Highly Selective and Orally Bioavailable Pim Kinases Inhibitors
Tao, Z.F., Hasvold, L., Leverson, J., Han, E., Guan, R., Johson, E.F., Stoll, V.S., Stewart, K.D., Stamper, G., Soni, N.
TO BE PUBLISHED
HeaderTransferase
Released2009-09-21
Resolution2.100
CATH Insert Date15 Nov, 2009

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 15 Nov, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3jyaA01 10 Apr, 2010 3.30.200.20 Assigned
3jyaA02 10 Apr, 2010 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1