PDB Information

PDB3IDP
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Selective inhibitors of the mutant B-raf pathway: discovery of a potent and orally bioavailable aminoisoquinoline.
Smith, A.L., Demorin, F.F., Paras, N.A., Huang, Q., Petkus, J.K., Doherty, E.M., Nixey, T., Kim, J.L., Whittington, D.A., Epstein, L.F., Lee, M.R., Rose, M.J., Babij, C., Fernando, M., Hess, K., Le, Q., Beltran, P., Carnahan, J.
J.Med.Chem.
HeaderTransferase
Released2009-07-21
Resolution2.700
CATH Insert Date08 Oct, 2009

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 09 Oct, 2009 Chopped
B 09 Oct, 2009 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3idpA01 28 Mar, 2010 3.30.200.20 Assigned
3idpA02 28 Mar, 2010 1.10.510.10 Assigned
3idpB01 28 Mar, 2010 3.30.200.20 Assigned
3idpB02 28 Mar, 2010 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf