PDB Information

PDB3ELM
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of potent, selective, and orally active carboxylic acid based inhibitors of matrix metalloproteinase-13
Monovich, L.G., Tommasi, R.A., Fujimoto, R.A., Blancuzzi, V., Clark, K., Cornell, W.D., Doti, R., Doughty, J., Fang, J., Farley, D., Fitt, J., Ganu, V., Goldberg, R., Goldstein, R., Lavoie, S., Kulathila, R., Macchia, W., Parker, D.T., Melton, R., O'Byrne, E., Pastor, G., Pellas, T., Quadros, E., Reel, N., Roland, D.M., Sakane, Y., Singh, H., Skiles, J., Somers, J., Toscano, K., Wigg, A., Zhou, S., Zhu, L., Shieh, W.C., Xue, S., McQuire, L.W.
J.Med.Chem.
HeaderHydrolase
Released2008-09-22
Resolution1.900
CATH Insert Date16 Aug, 2009

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2009 Chopped
B 16 Aug, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3elmA00 18 Mar, 2011 3.40.390.10 Assigned
3elmB00 18 Mar, 2011 3.40.390.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P45452 MMP13_HUMAN Homo sapiens Collagenase 3
P45452 MMP13_HUMAN Homo sapiens Collagenase 3