PDB Information

PDB3DPD
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Achieving multi-isoform PI3K inhibition in a series of substituted 3,4-dihydro-2H-benzo[1,4]oxazines
Perry, B., Alexander, R., Bennett, G., Buckley, G., Ceska, T., Crabbe, T., Dale, V., Gowers, L., Horsley, H., James, L., Jenkins, K., Crepy, K., Kulisa, C., Lightfoot, H., Lock, C., Mack, S., Morgan, T., Nicolas, A.-L., Pitt, W., Sabin, V., Wright, S.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-07-08
Resolution2.850
CATH Insert Date28 Aug, 2008

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Aug, 2008 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
3dpdA01 29 Aug, 2008 3.10.20.90 Assigned
3dpdA02 29 Aug, 2008 2.60.40.150 Assigned
3dpdA03 29 Aug, 2008 1.25.40.70 Assigned
3dpdA04 29 Aug, 2008 3.30.1010.10 Assigned
3dpdA05 29 Aug, 2008 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform