PDB Information

PDB3DD1
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Anthranilimide based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes. Part 3: X-ray crystallographic characterization, core and urea optimization and in vivo efficacy.
Thomson, S.A., Banker, P., Bickett, D.M., Boucheron, J.A., Carter, H.L., Clancy, D.C., Cooper, J.P., Dickerson, S.H., Garrido, D.M., Nolte, R.T., Peat, A.J., Sheckler, L.R., Sparks, S.M., Tavares, F.X., Wang, L., Wang, T.Y., Weiel, J.E.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-06-04
Resolution2.570
CATH Insert Date16 Aug, 2009

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2009 Chopped
B 16 Aug, 2009 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3dd1A01 15 Sep, 2009 3.40.50.2000 Assigned
3dd1A02 15 Sep, 2009 3.40.50.2000 Assigned
3dd1B01 15 Sep, 2009 3.40.50.2000 Assigned
3dd1B02 15 Sep, 2009 3.40.50.2000 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P06737 PYGL_HUMAN Homo sapiens Glycogen phosphorylase, liver form
P06737 PYGL_HUMAN Homo sapiens Glycogen phosphorylase, liver form