PDB Information

PDB3D0E
MethodX-RAY DIFFRACTION
Host Organismspodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Identification of 4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-{[(3S)-3-piperidinylmethyl]oxy}-1H-imidazo[4,5-c]pyridin-4-yl)-2-methyl-3-butyn-2-ol (GSK690693), a novel inhibitor of AKT kinase.
Heerding, D.A., Rhodes, N., Leber, J.D., Clark, T.J., Keenan, R.M., Lafrance, L.V., Li, M., Safonov, I.G., Takata, D.T., Venslavsky, J.W., Yamashita, D.S., Choudhry, A.E., Copeland, R.A., Lai, Z., Schaber, M.D., Tummino, P.J., Strum, S.L., Wood, E.R., Duckett, D.R., Eberwein, D., Knick, V.B., Lansing, T.J., McConnell, R.T., Zhang, S., Minthorn, E.A., Concha, N.O., Warren, G.L., Kumar, R.
J.Med.Chem.
HeaderTransferase Inhibitor
Released2008-05-01
Resolution2.000
CATH Insert Date23 Oct, 2008

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 23 Oct, 2008 Chopped
B 23 Oct, 2008 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3d0eA01 25 Oct, 2008 3.30.200.20 Assigned
3d0eA02 25 Oct, 2008 1.10.510.10 Assigned
3d0eB01 25 Oct, 2008 3.30.200.20 Assigned
3d0eB02 25 Oct, 2008 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P31751 AKT2_HUMAN Homo sapiens RAC-beta serine/threonine-protein kinase
P31751 AKT2_HUMAN Homo sapiens RAC-beta serine/threonine-protein kinase