PDB Information

PDB3CCN
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and Optimization of Triazolopyridazines as Potent and Selective Inhibitors of the c-Met Kinase.
Albrecht, B.K., Harmange, J.C., Bauer, D., Berry, L., Bode, C., Boezio, A.A., Chen, A., Choquette, D., Dussault, I., Fridrich, C., Hirai, S., Hoffman, D., Larrow, J.F., Kaplan-Lefko, P., Lin, J., Lohman, J., Long, A.M., Moriguchi, J., O'Connor, A., Potashman, M.H., Reese, M., Rex, K., Siegmund, A., Shah, K., Shimanovich, R., Springer, S.K., Teffera, Y., Yang, Y., Zhang, Y., Bellon, S.F.
J.Med.Chem.
HeaderTransferase
Released2008-02-26
Resolution1.900
CATH Insert Date01 May, 2008

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 01 May, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3ccnA01 10 Sep, 2008 3.30.200.20 Assigned
3ccnA02 10 Sep, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P08581 MET_HUMAN Homo sapiens Hepatocyte growth factor receptor