PDB Information

PDB2XYN
MethodX-RAY DIFFRACTION
Host OrganismTRICHOPLUSIA NI
Gene SourceHOMO SAPIENS
Primary Citation
Crystal Structures of Abl-Related Gene (Abl2) in Complex with Imatinib, Tozasertib (Vx-680), and a Type I Inhibitor of the Triazole Carbothioamide Class.
Salah, E., Ugochukwu, E., Barr, A.J., von Delft, F., Knapp, S., Elkins, J.M.
J.Med.Chem.
HeaderTransferase
Released2010-11-18
Resolution2.810
CATH Insert Date23 Jan, 2011

PDB Images (10)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 24 Jan, 2011 Chopped
B 24 Jan, 2011 Chopped
C 24 Jan, 2011 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
2xynA01 17 Feb, 2011 3.30.200.20 Assigned
2xynA02 17 Feb, 2011 1.10.510.10 Assigned
2xynB01 17 Feb, 2011 3.30.200.20 Assigned
2xynB02 17 Feb, 2011 1.10.510.10 Assigned
2xynC01 17 Feb, 2011 3.30.200.20 Assigned
2xynC02 17 Feb, 2011 1.10.510.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P42684 ABL2_HUMAN Homo sapiens Tyrosine-protein kinase ABL2
P42684 ABL2_HUMAN Homo sapiens Tyrosine-protein kinase ABL2
P42684 ABL2_HUMAN Homo sapiens Tyrosine-protein kinase ABL2