PDB Information

PDB2RL5
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Novel 2,3-dihydro-1,4-benzoxazines as potent and orally bioavailable inhibitors of tumor-driven angiogenesis.
La, D.S., Belzile, J., Bready, J.V., Coxon, A., Demelfi, T., Doerr, N., Estrada, J., Flynn, J.C., Flynn, S.R., Graceffa, R.F., Harriman, S.P., Larrow, J.F., Long, A.M., Martin, M.W., Morrison, M.J., Patel, V.F., Roveto, P.M., Wang, L., Weiss, M.M., Whittington, D.A., Teffera, Y., Zhao, Z., Polverino, A.J., Harmange, J.C.
J.Med.Chem.
HeaderTransferase
Released2007-10-18
Resolution2.650
CATH Insert Date10 Apr, 2008

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 Apr, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2rl5A01 10 Sep, 2008 3.30.200.20 Assigned
2rl5A02 10 Sep, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P35968 VGFR2_HUMAN Homo sapiens Vascular endothelial growth factor receptor 2