PDB Information

PDB2R7B
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Dibenzo[c,f][2,7]naphthyridines as Potent and Selective 3-Phosphoinositide-Dependent Kinase-1 Inhibitors.
Gopalsamy, A., Shi, M., Boschelli, D.H., Williamson, R., Olland, A.M., Hu, Y., Krishnamurthy, G., Han, X., Arndt, K., Guo, B.
J.Med.Chem.
HeaderSignaling Protein, Transferase
Released2007-09-07
Resolution2.700
CATH Insert Date11 Sep, 2008

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 11 Sep, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2r7bA01 12 Sep, 2008 3.30.200.20 Assigned
2r7bA02 12 Sep, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O15530 PDPK1_HUMAN Homo sapiens 3-phosphoinositide-dependent protein kinase 1