PDB Information

PDB2R4B
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
6-Ethynylthieno[3,2-d]- and 6-ethynylthieno[2,3-d]pyrimidin-4-anilines as tunable covalent modifiers of ErbB kinases.
Wood, E.R., Shewchuk, L.M., Ellis, B., Brignola, P., Brashear, R.L., Caferro, T.R., Dickerson, S.H., Dickson, H.D., Donaldson, K.H., Gaul, M., Griffin, R.J., Hassell, A.M., Keith, B., Mullin, R., Petrov, K.G., Reno, M.J., Rusnak, D.W., Tadepalli, S.M., Ulrich, J.C., Wagner, C.D., Vanderwall, D.E., Waterson, A.G., Williams, J.D., White, W.L., Uehling, D.E.
Proc.Natl.Acad.Sci.Usa
HeaderTransferase
Released2007-08-31
Resolution2.400
CATH Insert Date20 Mar, 2008

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 20 Mar, 2008 Chopped
B 20 Mar, 2008 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
2r4bA01 08 Dec, 2008 3.30.200.20 Assigned
2r4bA02 08 Dec, 2008 1.10.510.10 Assigned
2r4bB01 08 Dec, 2008 3.30.200.20 Assigned
2r4bB02 08 Dec, 2008 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q15303 ERBB4_HUMAN Homo sapiens Receptor tyrosine-protein kinase erbB-4
Q15303 ERBB4_HUMAN Homo sapiens Receptor tyrosine-protein kinase erbB-4