PDB Information

PDB2I47
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Identification of potent and selective TACE inhibitors via the S1 pocket.
Condon, J.S., Joseph-McCarthy, D., Levin, J.I., Lombart, H.G., Lovering, F.E., Sun, L., Wang, W., Xu, W., Zhang, Y.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2006-08-21
Resolution1.900
CATH Insert Date09 Jan, 2007

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2007 Chopped
B 09 Jan, 2007 Chopped
C 09 Jan, 2007 Chopped
D 09 Jan, 2007 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
2i47A00 10 Jan, 2007 3.40.390.10 Assigned
2i47B00 11 Jan, 2007 3.40.390.10 Assigned
2i47C00 11 Jan, 2007 3.40.390.10 Assigned
2i47D00 10 Jan, 2007 3.40.390.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17