PDB Information

PDB2GQG
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
The Structure of Dasatinib (BMS-354825) Bound to Activated ABL Kinase Domain Elucidates Its Inhibitory Activity against Imatinib-Resistant ABL Mutants
Tokarski, J.S., Newitt, J., Chang, C.Y.J., Cheng, J.D., Wittekind, M., Kiefer, S.E., Kish, K., Lee, F.Y.F., Borzilerri, R., Lombardo, L.J., Xie, D., Zhang, Y., Klei, H.E.
CANCER RES.
HeaderTransferase
Released2006-04-20
Resolution2.400
CATH Insert Date23 Nov, 2006

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 23 Nov, 2006 Chopped
B 23 Nov, 2006 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
2gqgA01 08 Dec, 2008 3.30.200.20 Assigned
2gqgA02 08 Dec, 2008 1.10.510.10 Assigned
2gqgB01 08 Dec, 2008 3.30.200.20 Assigned
2gqgB02 08 Dec, 2008 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1