PDB Information

PDB2C6E
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Sar and Inhibitor Complex Structure Determination of a Novel Class of Potent and Specific Aurora Kinase Inhibitors.
Heron, N.M., Anderson, M., Blowers, D.P., Breed, J., Eden, J.M., Green, S., Hill, G.B., Johnson, T., Jung, F.H., Mcmiken, H.H.J., Mortlock, A.A., Pannifer, A.D., Pauptit, R.A., Pink, J., Roberts, N.J., Rowsell, S.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Inhibitor
Released2005-11-09
Resolution2.100
CATH Insert Date05 Mar, 2006

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
2c6eA01 15 Mar, 2006 3.30.200.20 Assigned
2c6eA02 15 Mar, 2006 1.10.510.10 Assigned
2c6eB01 15 Mar, 2006 3.30.200.20 Assigned
2c6eB02 15 Mar, 2006 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O14965 AURKA_HUMAN Homo sapiens Aurora kinase A
O14965 AURKA_HUMAN Homo sapiens Aurora kinase A