CATH Domain 5kj0A01

CATH Classification

Level	CATH Code	Description
	1	Mainly Alpha
	1.20	Up-down Bundle
	1.20.920	Histone Acetyltransferase; Chain A
	1.20.920.10	Bromodomain-like

Domain Context

CATH Clusters

Superfamily	Bromodomain-like
Functional Family	Bromodomain-containing protein 4

Enzyme Information

UniProtKB Entries (1)

BRD4_HUMAN

Homo sapiens

Bromodomain-containing protein 4

PDB Structure

PDB	5KJ0
External Links	PDBSum Proteopedia
Method	X-RAY DIFFRACTION
Organism
Primary Citation	Assessment of Bromodomain Target Engagement by a Series of BI2536 Analogues with Miniaturized BET-BRET. Koblan, L.W., Buckley, D.L., Ott, C.J., Fitzgerald, M.E., Ember, S.W., Zhu, J.Y., Liu, S., Roberts, J.M., Remillard, D., Vittori, S., Zhang, W., Schonbrunn, E., Bradner, J.E. ChemMedChem