Discovery of PF-06928215 as a high affinity inhibitor of cGAS enabled by a novel fluorescence polarization assay.
Hall, J., Brault, A., Vincent, F., Weng, S., Wang, H., Dumlao, D., Aulabaugh, A., Aivazian, D., Castro, D., Chen, M., Culp, J., Dower, K., Gardner, J., Hawrylik, S., Golenbock, D., Hepworth, D., Horn, M., Jones, L., Jones, P., Latz, E., Li, J., Lin, L.L., Lin, W., Lin, D., Lovering, F., Niljanskul, N., Nistler, R., Pierce, B., Plotnikova, O., Schmitt, D., Shanker, S., Smith, J., Snyder, W., Subashi, T., Trujillo, J., Tyminski, E., Wang, G., Wong, J., Lefker, B., Dakin, L., Leach, K.
PLoS ONE
