CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Estrogen receptor

Enzyme Information

UniProtKB Entries (1)

P03372
ESR1_HUMAN
Homo sapiens
Estrogen receptor

PDB Structure

PDB 4ZN9
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Development of selective estrogen receptor modulator (SERM)-like activity through an indirect mechanism of estrogen receptor antagonism: defining the binding mode of 7-oxabicyclo[2.2.1]hept-5-ene scaffold core ligands.
Zheng, Y., Zhu, M., Srinivasan, S., Nwachukwu, J.C., Cavett, V., Min, J., Carlson, K.E., Wang, P., Dong, C., Katzenellenbogen, J.A., Nettles, K.W., Zhou, H.B.
Chemmedchem
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