PDB Information

PDB6UFX
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and Structure-Based Optimization of Potent and Selective WD repeat domain 5 (WDR5) Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core.
Tian, J., Teuscher, K., Aho, E.R., Alvarado, J.R., Mills, J.J., Meyers, K.M., Gogliotti, R.D., Han, C., Macdonald, J.D., Sai, J., Shaw, J.G., Sensintaffar, J.L., Zhao, B., Rietz, T.A., Thomas, L.R., Payne, W.G., Moore, W.J., Stott, G.M., Kondo, J., Inoue, M., Coffey, R., Tansey, W.P., Stauffer, S., Lee, T., Fesik, S.W.
J.Med.Chem.
HeaderGene Regulation/Inhibitor
Released2019-09-25
Resolution2.020
CATH Insert Date05 Jan, 2020

PDB Images (1)

PDB Prints

PDB Chains (0)

Chain ID Date inserted into CATH CATH Status

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (0)

Accession Gene ID Taxon Description