PDB 5zqq

PDB Information

PDB5ZQQ
MethodX-RAY DIFFRACTION
Host OrganismCell-free synthesis
Gene SourceHomo sapiens
Primary Citation
Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors.
Shirai, F., Tsumura, T., Yashiroda, Y., Yuki, H., Niwa, H., Sato, S., Chikada, T., Koda, Y., Washizuka, K., Yoshimoto, N., Abe, M., Onuki, T., Mazaki, Y., Hirama, C., Fukami, T., Watanabe, H., Honma, T., Umehara, T., Shirouzu, M., Okue, M., Kano, Y., Watanabe, T., Kitamura, K., Shitara, E., Muramatsu, Y., Yoshida, H., Mizutani, A., Seimiya, H., Yoshida, M., Koyama, H.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2018-04-19
Resolution2.290
CATH Insert Date07 Apr, 2019

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Apr, 2019 Chopped
B 07 Apr, 2019 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5zqqA00 08 Apr, 2019 3.90.228.10 Assigned
5zqqB00 08 Apr, 2019 6.20.320.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
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