PDB Information

PDB5TEG
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Turning a Substrate Peptide into a Potent Inhibitor for the Histone Methyltransferase SETD8.
Judge, R.A., Zhu, H., Upadhyay, A.K., Bodelle, P.M., Hutchins, C.W., Torrent, M., Marin, V.L., Yu, W., Vedadi, M., Li, F., Brown, P.J., Pappano, W.N., Sun, C., Petros, A.M.
ACS Med Chem Lett
HeaderTransferase
Released2016-09-21
Resolution1.300
CATH Insert Date08 Jan, 2017

PDB Images (7)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2017 Chopped
B 09 Jan, 2017 Chopped
D 09 Jan, 2017 Rejected
E 09 Jan, 2017 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5tegA00 16 Feb, 2017 2.170.270.10 Assigned
5tegB00 16 Feb, 2017 2.170.270.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P62805 H4_HUMAN Homo sapiens Histone H4
Q9NQR1 KMT5A_HUMAN Homo sapiens N-lysine methyltransferase KMT5A
P62805 H4_HUMAN Homo sapiens Histone H4
Q9NQR1 KMT5A_HUMAN Homo sapiens N-lysine methyltransferase KMT5A