PDB 5qik

PDB Information

PDB5QIK
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHomo sapiens
Primary Citation
Discovery of 4-Azaindole Inhibitors of TGF beta RI as Immuno-oncology Agents.
Zhang, Y., Zhao, Y., Tebben, A.J., Sheriff, S., Ruzanov, M., Fereshteh, M.P., Fan, Y., Lippy, J., Swanson, J., Ho, C.P., Wautlet, B.S., Rose, A., Parrish, K., Yang, Z., Donnell, A.F., Zhang, L., Fink, B.E., Vite, G.D., Augustine-Rauch, K., Fargnoli, J., Borzilleri, R.M.
ACS Med Chem Lett
HeaderTransferase/Transferase Inhibitor
Released2018-08-05
Resolution1.580
CATH Insert Date16 Dec, 2018

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5qikA01 28 Feb, 2019 3.30.200.20 Assigned
5qikA02 28 Feb, 2019 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P36897 TGFR1_HUMAN Homo sapiens TGF-beta receptor type-1