PDB Information

PDB5MG2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains.
Bouche, L., Christ, C.D., Siegel, S., Fernandez-Montalvan, A.E., Holton, S.J., Fedorov, O., Ter Laak, A., Sugawara, T., Stockigt, D., Tallant, C., Bennett, J., Monteiro, O., Diaz-Saez, L., Siejka, P., Meier, J., Putter, V., Weiske, J., Muller, S., Huber, K.V.M., Hartung, I.V., Haendler, B.
J. Med. Chem.
HeaderTranscription
Released2016-11-20
Resolution1.750
CATH Insert Date14 May, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 15 May, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5mg2A00 06 Nov, 2017 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P21675 TAF1_HUMAN Homo sapiens Transcription initiation factor TFIID subunit 1
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