PDB Information

PDB5LWM
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Selective JAK3 Inhibitors with a Covalent Reversible Binding Mode Targeting a New Induced Fit Binding Pocket.
Forster, M., Chaikuad, A., Bauer, S.M., Holstein, J., Robers, M.B., Corona, C.R., Gehringer, M., Pfaffenrot, E., Ghoreschi, K., Knapp, S., Laufer, S.A.
Cell Chem Biol
HeaderTransferase
Released2016-09-18
Resolution1.550
CATH Insert Date20 Nov, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 21 Nov, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5lwmA01 25 Nov, 2016 3.30.200.20 Assigned
5lwmA02 25 Nov, 2016 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P52333 JAK3_HUMAN Homo sapiens Tyrosine-protein kinase JAK3