Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours.
Lasko, L.M., Jakob, C.G., Edalji, R.P., Qiu, W., Montgomery, D., Digiammarino, E.L., Hansen, T.M., Risi, R.M., Frey, R., Manaves, V., Shaw, B., Algire, M., Hessler, P., Lam, L.T., Uziel, T., Faivre, E., Ferguson, D., Buchanan, F.G., Martin, R.L., Torrent, M., Chiang, G.G., Karukurichi, K., Langston, J.W., Weinert, B.T., Choudhary, C., de Vries, P., Van Drie, J.H., McElligott, D., Kesicki, E., Marmorstein, R., Sun, C., Cole, P.A., Rosenberg, S.H., Michaelides, M.R., Lai, A., Bromberg, K.D.
Nature
