Discovery of a Chemical Probe Bisamide (CCT251236): An Orally Bioavailable Efficacious Pirin Ligand from a Heat Shock Transcription Factor 1 (HSF1) Phenotypic Screen.
Cheeseman, M.D., Chessum, N.E., Rye, C.S., Pasqua, A.E., Tucker, M.J., Wilding, B., Evans, L.E., Lepri, S., Richards, M., Sharp, S.Y., Ali, S., Rowlands, M., O'Fee, L., Miah, A., Hayes, A., Henley, A.T., Powers, M., Te Poele, R., De Billy, E., Pellegrino, L., Raynaud, F., Burke, R., van Montfort, R.L., Eccles, S.A., Workman, P., Jones, K.
J. Med. Chem.
