PDB 4rg0
PDB Information
PDB | 4RG0 |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | Finding the perfect spot for fluorine: Improving potency up to 40-fold during a rational fluorine scan of a Bruton's Tyrosine Kinase (BTK) inhibitor scaffold.
Bioorg.Med.Chem.Lett.
|
Header | Transferase/Transferase Inhibitor |
Released | 2014-09-29 |
Resolution | 2.500 |
CATH Insert Date | 04 Jan, 2015 |
PDB Images (4)
PDB Prints
PDB Chains (1)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 05 Jan, 2015 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4rg0A01 | 10 Jan, 2015 | 3.30.200.20 | Assigned |
4rg0A02 | 10 Jan, 2015 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q06187 | BTK_HUMAN | Homo sapiens | Tyrosine-protein kinase BTK |