PDB 4qr3

PDB Information

PDB4QR3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Fragment-based drug discovery of 2-thiazolidinones as BRD4 inhibitors: 2. Structure-based optimization
Zhao, L., Wang, Y., Cao, D.Y., Chen, T.T., Wang, Q., Li, Y., Xu, Y.C., Zhang, N., Wang, X., Chen, D., Chen, L., Chen, Y.L., Xia, G., Shi, Z., Liu, Y.C., Lin, Y., Miao, Z., Shen, J., Xiong, B.
J.Med.Chem.
HeaderTranscription/Transcription Inhibitor
Released2014-06-30
Resolution1.370
CATH Insert Date16 Aug, 2015

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4qr3A01 24 Aug, 2015 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
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