PDB 4msk
PDB Information
PDB | 4MSK |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Development of novel dual binders as potent, selective, and orally bioavailable tankyrase inhibitors.
J.Med.Chem.
|
Header | Transferase/Transferase Inhibitor |
Released | 2013-09-18 |
Resolution | 2.300 |
CATH Insert Date | 05 Jan, 2014 |
PDB Images (9)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 06 Jan, 2014 | Chopped |
B | 06 Jan, 2014 | Chopped |
C | 06 Jan, 2014 | Chopped |
D | 06 Jan, 2014 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4mskA00 | 09 Jan, 2014 | 3.90.228.10 | Assigned |
4mskB00 | 09 Jan, 2014 | 3.90.228.10 | Assigned |
4mskC00 | 09 Jan, 2014 | 3.90.228.10 | Assigned |
4mskD00 | 09 Jan, 2014 | 3.90.228.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
O95271 | TNKS1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-1 |
O95271 | TNKS1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-1 |
O95271 | TNKS1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-1 |
O95271 | TNKS1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-1 |