PDB 4mr5

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PDB Links
Overview

PDB Information

PDB	4MR5
Method	X-RAY DIFFRACTION
Host Organism	Escherichia coli
Gene Source	Homo sapiens
Primary Citation	RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. Picaud, S., Wells, C., Felletar, I., Brotherton, D., Martin, S., Savitsky, P., Diez-Dacal, B., Philpott, M., Bountra, C., Lingard, H., Fedorov, O., Muller, S., Brennan, P.E., Knapp, S., Filippakopoulos, P. Proc.Natl.Acad.Sci.USA
Header	Transcription/Transcription Inhibitor
Released	2013-09-17
Resolution	1.630
CATH Insert Date	01 Dec, 2013

PDB Images (3)

Image of CATH 4mr5

4mr5

PDB 4mr5

Image of CATH 4mr5A

4mr5A

PDB Chain 4mr5A

Image of CATH 4mr5A00

4mr5A00

CATH Domain 4mr5A00

PDB Prints

PDB Chains (1)

Chain ID	Date inserted into CATH	CATH Status
A	02 Dec, 2013	Chopped

CATH Domains (1)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
4mr5A00	04 Dec, 2013	1.20.920.10	Assigned

UniProtKB Entries (1)

Accession	Gene ID	Taxon	Description
P25440	BRD2_HUMAN	Homo sapiens	Bromodomain-containing protein 2