PDB 4lrg

PDB Information

PDB4LRG
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors.
Gehling, V.S., Hewitt, M.C., Vaswani, R.G., Leblanc, Y., Cote, A., Nasveschuk, C.G., Taylor, A.M., Harmange, J.C., Audia, J.E., Pardo, E., Joshi, S., Sandy, P., Mertz, J.A., Sims, R.J., Bergeron, L., Bryant, B.M., Bellon, S., Poy, F., Jayaram, H., Sankaranarayanan, R., Yellapantula, S., Bangalore Srinivasamurthy, N., Birudukota, S., Albrecht, B.K.
ACS Med Chem Lett
HeaderTranscription Regulator/Inhibitor
Released2013-07-19
Resolution2.210
CATH Insert Date01 Sep, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 02 Sep, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4lrgA01 03 Sep, 2013 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
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