PDB 4lr6

PDB Information

PDB4LR6
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors.
Gehling, V.S., Hewitt, M.C., Vaswani, R.G., Leblanc, Y., Cote, A., Nasveschuk, C.G., Taylor, A.M., Harmange, J.C., Audia, J.E., Pardo, E., Joshi, S., Sandy, P., Mertz, J.A., Sims, R.J., Bergeron, L., Bryant, B.M., Bellon, S., Poy, F., Jayaram, H., Sankaranarayanan, R., Yellapantula, S., Bangalore Srinivasamurthy, N., Birudukota, S., Albrecht, B.K.
ACS Med Chem Lett
HeaderTranscription Regulator/Inhibitor
Released2013-07-19
Resolution1.290
CATH Insert Date01 Sep, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 02 Sep, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4lr6A01 04 Sep, 2013 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
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