PDB 4geb
PDB Information
PDB | 4GEB |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | PF-04859989 as a template for structure-based drug design: identification of new pyrazole series of irreversible KAT II inhibitors with improved lipophilic efficiency.
Bioorg.Med.Chem.Lett.
|
Header | Transferase/Transferase Inhibitor |
Released | 2012-08-01 |
Resolution | 2.150 |
CATH Insert Date | 28 Mar, 2013 |
PDB Images (9)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 28 Mar, 2013 | Chopped |
B | 28 Mar, 2013 | Chopped |
CATH Domains (6)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4gebA01 | 30 Aug, 2013 | Holding pen | |
4gebA02 | 30 Aug, 2013 | 3.40.640.10 | Assigned |
4gebA03 | 30 Aug, 2013 | 3.90.1150.10 | Assigned |
4gebB01 | 30 Aug, 2013 | Holding pen | |
4gebB02 | 30 Aug, 2013 | 3.40.640.10 | Assigned |
4gebB03 | 30 Aug, 2013 | 3.90.1150.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q8N5Z0 | AADAT_HUMAN | Homo sapiens | Kynurenine/alpha-aminoadipate aminotransferase, mitochondrial |
Q8N5Z0 | AADAT_HUMAN | Homo sapiens | Kynurenine/alpha-aminoadipate aminotransferase, mitochondrial |