PDB 3sx0
PDB Information
PDB | 3SX0 |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Bromo-deaza-SAH: a potent and selective DOT1L inhibitor.
Bioorg. Med. Chem.
|
Header | Transferase |
Released | 2011-07-14 |
Resolution | 2.280 |
CATH Insert Date | 07 Aug, 2011 |
PDB Images (4)
PDB Prints
PDB Chains (1)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 08 Aug, 2011 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
3sx0A01 | 12 Aug, 2011 | 1.10.260.60 | Assigned |
3sx0A02 | 12 Aug, 2011 | 3.40.50.150 | Assigned |
UniProtKB Entries (1)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q8TEK3 | DOT1L_HUMAN | Homo sapiens | Histone-lysine N-methyltransferase, H3 lysine-79 specific |