PDB Information

PDB3P9J
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of aurora-a kinase.
Prime, M.E., Courtney, S.M., Brookfield, F.A., Marston, R.W., Walker, V., Warne, J., Boyd, A.E., Kairies, N.A., von der Saal, W., Limberg, A., Georges, G., Engh, R.A., Goller, B., Rueger, P., Rueth, M.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2010-10-17
Resolution2.800
CATH Insert Date27 Mar, 2011

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Mar, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3p9jA01 01 Apr, 2011 3.30.200.20 Assigned
3p9jA02 01 Apr, 2011 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14965 AURKA_HUMAN Homo sapiens Aurora kinase A
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