PDB Information

PDB2E9N
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of 1,4-dihydroindeno[1,2-c]pyrazoles as a novel class of potent and selective checkpoint kinase 1 inhibitors.
Tong, Y., Claiborne, A., Stewart, K.D., Park, C., Kovar, P., Chen, Z., Credo, R.B., Gu, W.Z., Gwaltney, S.L., Judge, R.A., Zhang, H., Rosenberg, S.H., Sham, H.L., Sowin, T.J., Lin, N.H.
Bioorg.Med.Chem.
HeaderTransferase
Released2007-01-26
Resolution2.500
CATH Insert Date21 Feb, 2008

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 21 Feb, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2e9nA01 23 Feb, 2008 3.30.200.20 Assigned
2e9nA02 23 Feb, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14757 CHK1_HUMAN Homo sapiens Serine/threonine-protein kinase Chk1
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