PDB 1x81
PDB Information
PDB | 1X81 |
Method | X-RAY DIFFRACTION |
Host Organism | |
Gene Source | |
Primary Citation | Design, synthesis, and activity of 4-quinolone and pyridone compounds as nonthiol-containing farnesyltransferase inhibitors.
Bioorg.Med.Chem.Lett.
|
Header | Transferase |
Released | 2004-08-16 |
Resolution | 3.500 |
CATH Insert Date | 05 Mar, 2006 |
PDB Images (5)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 05 Mar, 2006 | Chopped |
B | 05 Mar, 2006 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
1x81A00 | 09 Mar, 2006 | 1.25.40.120 | Assigned |
1x81B00 | 09 Mar, 2006 | 1.50.10.20 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q04631 | FNTA_RAT | Rattus norvegicus | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
Q02293 | FNTB_RAT | Rattus norvegicus | Protein farnesyltransferase subunit beta |