PDB Information

PDB3DDS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Anthranilimide based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes. Part 3: X-ray crystallographic characterization, core and urea optimization and in vivo efficacy.
Thomson, S.A., Banker, P., Bickett, D.M., Boucheron, J.A., Carter, H.L., Clancy, D.C., Cooper, J.P., Dickerson, S.H., Garrido, D.M., Nolte, R.T., Peat, A.J., Sheckler, L.R., Sparks, S.M., Tavares, F.X., Wang, L., Wang, T.Y., Weiel, J.E.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-06-06
Resolution1.800
CATH Insert Date29 Jan, 2009

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jan, 2009 Chopped
B 29 Jan, 2009 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3ddsA01 18 Feb, 2009 3.40.50.2000 Assigned
3ddsA02 18 Feb, 2009 3.40.50.2000 Assigned
3ddsB01 19 Feb, 2009 3.40.50.2000 Assigned
3ddsB02 19 Feb, 2009 3.40.50.2000 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P06737 PYGL_HUMAN Homo sapiens Glycogen phosphorylase, liver form
P06737 PYGL_HUMAN Homo sapiens Glycogen phosphorylase, liver form